Kodi pali kusiyana kotani pakati pa mitundu inayi ya "paclitaxel"?

Paclitaxel, yomwe imadziwikanso kuti red paclitaxel,tamsulosin,violet,ndi tesu,ndi mankhwala abwino kwambiri achilengedwe othana ndi khansa omwe apezeka mpaka pano, ndipo amagwiritsidwa ntchito kwambiri pochiza khansa ya m'mawere, khansa ya m'mawere, khansa ya mutu ndi khosi. Khansara ya m'mapapo. Monga mankhwala amtundu wa chemotherapy, dzina lapaclitaxelakukhulupirira kuti anthu ambiri adamvapo.Tiyeni tiwone kusiyana kwa mitundu inayi ya paclitaxel m'nkhani yotsatirayi.

paclitaxel

Kusiyana kwa mitundu inayi yapaclitaxel

1, Paclitaxel: Imagwira pa microtubule/microtubule protein system, imaletsa kufooketsa kwa microtubule, imatchinga ma cell mu gawo la G2/M, imayambitsa mitosis kapena kumangidwa, imalepheretsa kuchulukana kwa maselo a khansa, ndikupanga maselo a khansa kulephera kupitilira kugawa ndi kufa.

2, Docetaxel: The limagwirira ntchito ndi chimodzimodzi ndi paclitaxel, koma ndi apamwamba kuyanjana kwa microtubule kumanga malo ndi apamwamba odana ndi khansa ntchito.

3, Liposomal paclitaxel: Liposomal paclitaxel: limagwirira ntchito ndi chimodzimodzi ndi paclitaxel. The liposomes wapangidwa lecithin, mafuta m`thupi, threonine ndi zipangizo zofanana ndi phospholipid bilayer dongosolo la cell nembanemba encapsulate paclitaxel, amene akhoza kusintha madzi solubility, kulowa mosavuta. kulowa m'mitsempha yamagazi, ndikuchepetsa kawopsedwe ka mtima ndi impso, ndi zina.

4.Albumin-bound paclitaxel:hydrophobic paclitaxel imaphatikizidwa ndi serum albumin carrier ndi nanotechnology.Albumin ikhoza kuwonjezera kutengeka kwa paclitaxel mu chotupa pomanga ku gp60 receptor ndikuwonjezera kuchuluka kwa paclitaxel mu minofu ya chotupa, motero kumawonjezera mphamvu yotsutsa-chotupa. .

Paclitaxel,doxorubicin,paclitaxel liposome kapena albumin paclitaxel ndi mtundu womwewo wa mankhwala a chemotherapeutic,ndipo onse ali mgulu la paclitaxel mgulu la mankhwala a chemotherapeutic.Ndi mankhwala amtundu womwewo.Paclitaxel ndi mankhwala oletsa kutupa omwe ali ndi mfundo ya microtubule inhibitor, yomwe imagwiritsidwa ntchito kwambiri pamankhwala a khansa ya m'mawere.

Zindikirani: Zomwe zingatheke komanso momwe mungagwiritsire ntchito ulalikiwu zimachokera m'mabuku osindikizidwa.

paclitaxel API

Kuwerenga kowonjezereka:Yunnan Hande Biotechnology Co., Ltd. yakhala ikuyang'ana kwambiri pakupanga paclitaxel kwa zaka 28.Ndiwodzipangira yekha padziko lonse lapansi wopanga mankhwala oletsa khansa a paclitaxel omwe avomerezedwa ndi US FDA, European EDQM, Australian TGA, China CFDA, India, Japan ndi mabungwe ena olamulira dziko.bizinesi.Ngati mukufuna kugulaPaclitaxel API, chonde titumizireni pa intaneti.


Nthawi yotumiza: Oct-08-2022