High Quality cabazitaxel mphamvu Cabazitaxel wopanga

Kufotokozera Kwachidule:

Carbataxel ndi mankhwala omwe amagwiritsidwa ntchito popanga mankhwala oletsa khansa.Carbataxel ndi ufa woyera kapena woyera womwe umakhala wosasungunuka m'madzi, koma umasungunuka mu ethanol.Njira yake yolimbana ndi khansa ndi mawonekedwe ake ndi ofanana ndi docetaxel, ndipo ali m'gulu la mankhwala odana ndi microtubule.Kudzera kuphatikiza ndi tubulin, kulimbikitsa ake kusonkhana mu microtubules, pa nthawi yomweyo zingalepheretse awa wasonkhana ndi microtubule disassembly, kuti bata microtubules, potero inhibiting selo mitosis, ndi interphase selo ntchito (interphasecellularfunctions).


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Zambiri Zamalonda

Dzina:Cabazitaxel

Nambala ya CAS:183133-96-2

Chemical formula:C45H57NO14

Zofotokozera:99%

Mtundu:ufa woyera kapena woyera

Gwero:Semi-synthesized ndi 10-DAB

Mtundu:APIs

Udindo ndi ubwino wa cabataxel

1.anti-cancer effect: carbamazel imakhala ndi mphamvu yotsutsa khansa, imatha kulepheretsa kukula ndi kufalikira kwa maselo otupa, kupangitsa kuti maselo a khansa apangidwe.Poyerekeza ndi chilengedwe cha paclitaxel, carbataxel ili ndi zochita zambiri zotsutsana ndi khansa komanso zotsutsana ndi khansa.

2.chitetezo: Cabataxel pakupanga ndi kupanga, yang'anani pakuwongolera chitetezo chazinthu ndi kulolerana.Mwa kusintha ndi kukhathamiritsa kapangidwe ka mankhwala a paclitaxel, kuchuluka kwa zotsatirapo zoyipa komanso zoyipa zidachepetsedwa.

3.pharmacokinetic makhalidwe: carbamazel ali ndi makhalidwe abwino a pharmacokinetic, kotero kuti akhoza kutengeka bwino ndi kugawidwa mu thupi, kuti apititse patsogolo chithandizo chamankhwala.

4.applicability: carbataxel ingagwiritsidwe ntchito pochiza mitundu yosiyanasiyana ya khansa, kuphatikizapo khansa ya m'mapapo, khansa ya m'mawere, khansara ya ovarian, khansa ya m'mimba, ndi zina zotero. Kuchita kwake ndi chitetezo zatsimikiziridwa kwambiri kuchipatala.

5.Thandizo la sayansi: Cabataxel imachokera ku kafukufuku waposachedwapa wa sayansi ndi chitukuko cha zamakono, ndi chithandizo chodalirika cha sayansi.

Ntchito Zathu

1.Zogulitsa:Perekani zokometsera zapamwamba kwambiri, zoyera kwambiri, zopangira mankhwala, komanso zopangira mankhwala.

2.Ntchito zaukadaulo:Makonda akupanga ndi specifications wapadera malinga ndi zofunika kasitomala.

Hande fakitale

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