Zambiri Zamalonda
Dihydroartemisinin ndi yochokera ku artemisinin, amene ali amphamvu ndi mofulumira kupha zotsatira pa erythrocytic gawo la malungo tiziromboti, ndipo mwamsanga kulamulira matenda kuukira ndi zizindikiro.
1, Gwero chomera
Dihydroartemisinin ndi chotumphukira cha artemisinin.Artemisinin ndi mankhwala oletsa malungo otengedwa ku Artemisia annua.
2. Udindo
The pharmacological zochita za dihydroartemisinin ndi ofanana ndi artemisinin.Zotsatira za artemisinin pa ultrastructure wa Plasmodium falciparum mu gawo erythrocytic makamaka kusintha nembanemba dongosolo.Mankhwalawa amayamba kugwira ntchito pa nembanemba ya vesicle ya chakudya, nembanemba ya pamwamba ndi mitochondria, kenako ndi nembanemba ya nyukiliya ndi endoplasmic reticulum.Kuphatikiza apo, imakhudzanso chromatin mu phata.Ikhoza kugwira ntchito pa nembanemba ya chakudya, kutsekereza siteji yoyambirira ya kudya kwa malungo, kuchititsa kuti tizilombo toyambitsa malungo tife msanga ndi njala ya ma amino acid, kupanga ma autophagic vesicles, ndi kutuluka m'thupi mosalekeza, kutaya kuchuluka kwa madzi. cytoplasm ndi zakudya, koma osati kuwonjezeredwa, choncho mwamsanga amafa.Kachitidwe ake makamaka kusokoneza ntchito ya Plasmodium pamwamba nembanemba mitochondria.Kupyolera mu mlatho wake wamkati wa peroxide (dioxygen), umalumikizidwa ndi chitsulo chaulere chomwe chimapangidwa pambuyo pa kuwonongeka kwa hemoglobin kuti apange ma radicals aulere osakhazikika komanso / kapena ma electrophilic intermediates, kenako amapanga ma covalent adducts ndi mapuloteni a malungo, zomwe zimapangitsa imfa ya tizilombo ta malungo.Kutenga kwa tritium yotchedwa isoleucine ndi cultured Plasmodium falciparum in vitro kunasonyezanso kuti njira yake yoyamba ingakhale yolepheretsa kaphatikizidwe ka mapuloteni a Plasmodium.
3. Munda wa ntchito
1. Makampani opanga mankhwala
Product Parameters
MBIRI YAKAMPANI | |
Dzina lazogulitsa | Dihydroartemisinin |
CAS | 81496-82-4 |
Chemical Formula | C15H24O5 |
Brandi | Hndi |
Mwopanga | YMalingaliro a kampani unnan Hande Bio-Tech Co., Ltd. |
Ckunja | Kunming,Cine |
Kukhazikitsidwa | 1993 |
BMALANGIZO ASIC | |
Mawu ofanana ndi mawu | (3R,5aS,6R,8aS,9R,12S,12aR) -octahydrogen -3,6,9-trimethyl -3,12-epoxy -12H-pyrane [4,3-j]-1,2-coumaron -10 ( 3H ) mowa;Dihydroartemisinin;Dihxdroarteannui;Dihydroartemisinin USP/EP/BP |
Kapangidwe | |
Kulemera | 284.35 |
HS kodi | N / A |
UbwinoStanthauzo | Mafotokozedwe a Kampani |
Czotsimikizira | N / A |
Kuyesa | Zosinthidwa malinga ndi zosowa za makasitomala |
Maonekedwe | Mwala woyera |
Njira Yochotsera | Artemisia annua Linn. |
Kutha Kwapachaka | Zosinthidwa malinga ndi zosowa za makasitomala |
Phukusi | Zosinthidwa malinga ndi zosowa za makasitomala |
Njira Yoyesera | Mtengo wa HPLC |
Kayendesedwe | Zambiritransports |
PayimentTerms | T/T, D/P, D/A |
Oawo | Landirani kuwunika kwamakasitomala nthawi zonse;Thandizani makasitomala polembetsa zowongolera. |
Hande product statement
1.Zogulitsa zonse zomwe zimagulitsidwa ndi kampaniyo ndi zopangira zomaliza.Zogulitsazo zimayang'ana makamaka kwa opanga omwe ali ndi ziyeneretso zopanga, ndipo zopangira sizinthu zomaliza.
2.Kuthekera kothekera ndi ntchito zomwe zikuphatikizidwa m'mawu oyamba onse amachokera m'mabuku osindikizidwa.Anthu samalimbikitsa kugwiritsa ntchito mwachindunji, ndipo kugula payekha kumakanidwa.
3. Zithunzi ndi zambiri zazinthu zomwe zili patsamba lino ndizongongotchula zokhazokha, ndipo zomwe zili zenizeni ndizoyenera.